Difference between revisions of "User:Etienne Robillard/Notebook/Drospirenone"

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* optical isomerism (C2) : a HSL (homoserine) lactone derivative ?
 
* optical isomerism (C2) : a HSL (homoserine) lactone derivative ?
 
* A high risks of hyperkalemia (K+) was found with long-term use of Yasmin. [http://sante.canoe.ca/drug_info_details.asp?brand_name_id=2052 2]
 
* A high risks of hyperkalemia (K+) was found with long-term use of Yasmin. [http://sante.canoe.ca/drug_info_details.asp?brand_name_id=2052 2]
* Ethics of birth control with chiral schiff base alkyloids in orthogonal Fmoc-carbonyl nucleophilic catalysis? See [http://en.wikipedia.org/wiki/Grignard_reagent Grignard reagent] .
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* Ethics of birth control with chiral Schiff base alkyloids in orthogonal Fmoc-carbonyl nucleophilic catalysis? See [http://en.wikipedia.org/wiki/Grignard_reagent Grignard reagent] .
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* Hence, is there a Yb(OTf)3 (distereoselective) route to remote activation of Fmoc-protected alkylamines via MW catalysis of C(2)-symmetric amines, ie Drospirenone ? See http://www.organic-chemistry.org/abstracts/literature/979.shtm
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== References ==
 
== References ==
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# http://en.wikipedia.org/wiki/Drospirenone
 
# http://en.wikipedia.org/wiki/Drospirenone
 
# http://en.wikipedia.org/wiki/Spironolactone
 
# http://en.wikipedia.org/wiki/Spironolactone
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== See also ==
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[[Pyrrolidines]]

Revision as of 08:45, 4 February 2013

  • CYP450 mediated [1] (A spironolactone derived alkyloid)
  • optical isomerism (C2) : a HSL (homoserine) lactone derivative ?
  • A high risks of hyperkalemia (K+) was found with long-term use of Yasmin. 2
  • Ethics of birth control with chiral Schiff base alkyloids in orthogonal Fmoc-carbonyl nucleophilic catalysis? See Grignard reagent .
  • Hence, is there a Yb(OTf)3 (distereoselective) route to remote activation of Fmoc-protected alkylamines via MW catalysis of C(2)-symmetric amines, ie Drospirenone ? See http://www.organic-chemistry.org/abstracts/literature/979.shtm


References

  1. http://en.wikipedia.org/wiki/Drospirenone
  2. http://en.wikipedia.org/wiki/Spironolactone

See also

Pyrrolidines